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Cat No. | Product Name | Synonyms | Targets |
---|---|---|---|
T11363 | Ganoderic acid F | Others | |
Ganoderic acid F exhibits antitumor and antimetastatic activities through inhibition of angiogenesis and alteration of proteins involving cell proliferation and/or cell death, carcinogenesis, oxidative stress, calcium si... | |||
T36816 | S-trityl-L-Cysteine | STLC | Kinesin |
S-trityl-L-Cysteine is a non-natural amino acid and an inhibitor of Eg5, also known as KSP and Kif11, a mitotic kinesin necessary for mitotic spindle formation. S-trityl-L-Cysteine inhibits the ATPase activity of Eg5 in ... | |||
T21685 | CCT 031374 hydrobromide | Wnt/beta-catenin | |
CCT 031374 hydrobromide is a TCF/β-catenin inhibitor with antitumor activities. | |||
T3389 | Antitumor agent-21 | TRX818 | Others |
Antitumor agent-21 (TRX818) is an orally bioavailable agent with potential antineoplastic and anti-vasculogenic mimicry (VM) activities. | |||
T9991 | WAY-620645 | cholecystokinin | |
WAY-620645 is a CCK antagonist with antitumor and analgesic activities. | |||
T9940 | Protein kinase G inhibitor-2 | Others | |
Protein kinase G inhibitor-2 exhibits antibacterial, antiviral, and antitumor activities. | |||
T19668 | Tiomolibdate diammonium | Ammonium molybdenum sulfide,Ammonium tetrathiomolybdate,NSC 286644,ATTM,Coprexa | Others |
Tiomolibdate diammonium (NSC-286644) is an inhibitor of superoxide dismutase 1 (SOD1) exerting antiangiogenic and antitumor activities. Tiomolibdate diammonium inhibits the activities of cuproenzymes, including SOD1 and ... | |||
T6473 | Dioscin | CCRIS 4123,Collettiside III,Saponin | Apoptosis , Autophagy |
Dioscin (Collettiside III) is a saponin with antitumor activities. | |||
T14885 | CBS9106 | SL-801 | CRM1 |
CBS9106 (SL-801) is a reversible oral inhibitor of CRM1 with CRM1 degrading and antitumor activities. CBS9106 arrests the cell cycle and inducing apoptosis in a time- and dose-dependent manner for a broad spectrum of can... | |||
T1898 | RKI-1447 | RKI1447 | ROCK |
RKI-1447 is a potent inhibitor of ROCK1 and ROCK2. It has anti-invasive and antitumor activities. | |||
T9399 | Menin-MLL inhibitor 20 | Epigenetic Reader Domain , Histone Methyltransferase | |
Menin-MLL inhibitor 20 is an irreversible inhibitor of menin-MLL interaction with antitumor activities. | |||
T3819 | Ursolic acid acetate | Acetylursolic acid,3-Acetylursolic Acid | AChE |
Ursolic acid acetate (Acetylursolic acid) has cytotoxic activity, antimalarial activity, antitumor and anticancer activities. Acetylursolic acid has NO production inhibitory activities. Acetylursolic acid has inhibition ... | |||
T9999 | Sirtuin modulator 2 | N-(3-(imidazo[2,1-b]thiazol-6-yl)phenyl)-2-methoxybenzamide | Others , Sirtuin |
Sirtuin modulator 2 (N-(3-(imidazo[2,1-b]thiazol-6-yl)phenyl)-2-methoxybenzamide) exhibits antidiabetic, anti-inflammatory and antitumor activities. | |||
T0707 | Cyclophosphamide hydrate | Cyclophosphamide monohydrate | DNA Alkylator/Crosslinker , DNA , MRP |
Cyclophosphamide hydrate is a DNA alkylating agent, an inhibitor of DNA synthesis. Cyclophosphamide hydrate has antitumor and immunosuppressive activities. | |||
T2863 | P-Coumaric acid | para-Coumaric Acid,4-Hydroxycinnamic acid,trans-4-Hydroxycinnamic acid,Trans-p-Coumaric acid,4-Coumaric acid,P-Hydroxycinnamic acid | Endogenous Metabolite , Antibiotic |
p-Coumaric acid (para-Coumaric Acid) is the abundant isomer of cinnamic acid, with antitumor and anti-mutagenic activities. | |||
T2997 | Rhein | Rheinic Acid,Monorhein,NSC 38629,Rheic Acid,Rhubarb yellow | Reactive Oxygen Species , Antibacterial , Autophagy |
Rhein (NSC 38629) is an anthraquinone compound extracted from Polygonaceae Rheum Officinale with anti-inflammation and antitumor activities. | |||
TN1190 | 14,15 β-Dihydroxyklaineanone | 14,15beta-Dihydroxyklaineanone | Parasite |
14,15 β-Dihydroxyklaineanone(14,15beta-Dihydroxyklaineanone) is a bittersweet compound isolated from Eurycoma longifolia with antitumor-promoting, antischistosomal and plasmodium-killing activities. | |||
T2853 | Curcumol | (-)-Curcumol | Apoptosis , JAK |
Curcumol ((-)-Curcumol), a pure monomer isolated extracted from Rhizoma Curcumaeis, has antitumor activities. | |||
T7470 | 6-Chloropurine | 6-Chloro-9H-purine | Others |
6-Chloropurine (6-Chloro-9H-purine) is a building block in chemical synthesis,with Antitumor activities. | |||
T0876 | Clioquinol | Chinoform,Iodochlorhydroxyquin | Mitophagy , Antibiotic , Autophagy , Antifungal |
Clioquinol (Iodochlorhydroxyquin) is an orally bioavailable, lipophilic, copper-binding, halogenated 8-hydroxyquinoline with antifungal, antiparasitic and potential antitumor activities. |