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Search Results for " antitumor activities "

20

Compounds

Cat No. Product Name Synonyms Targets
T11363 Ganoderic acid F Others
Ganoderic acid F exhibits antitumor and antimetastatic activities through inhibition of angiogenesis and alteration of proteins involving cell proliferation and/or cell death, carcinogenesis, oxidative stress, calcium si...
T36816 S-trityl-L-Cysteine STLC Kinesin
S-trityl-L-Cysteine is a non-natural amino acid and an inhibitor of Eg5, also known as KSP and Kif11, a mitotic kinesin necessary for mitotic spindle formation. S-trityl-L-Cysteine inhibits the ATPase activity of Eg5 in ...
T21685 CCT 031374 hydrobromide Wnt/beta-catenin
CCT 031374 hydrobromide is a TCF/β-catenin inhibitor with antitumor activities.
T3389 Antitumor agent-21 TRX818 Others
Antitumor agent-21 (TRX818) is an orally bioavailable agent with potential antineoplastic and anti-vasculogenic mimicry (VM) activities.
T9991 WAY-620645 cholecystokinin
WAY-620645 is a CCK antagonist with antitumor and analgesic activities.
T9940 Protein kinase G inhibitor-2 Others
Protein kinase G inhibitor-2 exhibits antibacterial, antiviral, and antitumor activities.
T19668 Tiomolibdate diammonium Ammonium molybdenum sulfide,Ammonium tetrathiomolybdate,NSC 286644,ATTM,Coprexa Others
Tiomolibdate diammonium (NSC-286644) is an inhibitor of superoxide dismutase 1 (SOD1) exerting antiangiogenic and antitumor activities. Tiomolibdate diammonium inhibits the activities of cuproenzymes, including SOD1 and ...
T6473 Dioscin CCRIS 4123,Collettiside III,Saponin Apoptosis , Autophagy
Dioscin (Collettiside III) is a saponin with antitumor activities.
T14885 CBS9106 SL-801 CRM1
CBS9106 (SL-801) is a reversible oral inhibitor of CRM1 with CRM1 degrading and antitumor activities. CBS9106 arrests the cell cycle and inducing apoptosis in a time- and dose-dependent manner for a broad spectrum of can...
T1898 RKI-1447 RKI1447 ROCK
RKI-1447 is a potent inhibitor of ROCK1 and ROCK2. It has anti-invasive and antitumor activities.
T9399 Menin-MLL inhibitor 20 Epigenetic Reader Domain , Histone Methyltransferase
Menin-MLL inhibitor 20 is an irreversible inhibitor of menin-MLL interaction with antitumor activities.
T3819 Ursolic acid acetate Acetylursolic acid,3-Acetylursolic Acid AChE
Ursolic acid acetate (Acetylursolic acid) has cytotoxic activity, antimalarial activity, antitumor and anticancer activities. Acetylursolic acid has NO production inhibitory activities. Acetylursolic acid has inhibition ...
T9999 Sirtuin modulator 2 N-(3-(imidazo[2,1-b]thiazol-6-yl)phenyl)-2-methoxybenzamide Others , Sirtuin
Sirtuin modulator 2 (N-(3-(imidazo[2,1-b]thiazol-6-yl)phenyl)-2-methoxybenzamide) exhibits antidiabetic, anti-inflammatory and antitumor activities.
T0707 Cyclophosphamide hydrate Cyclophosphamide monohydrate DNA Alkylator/Crosslinker , DNA , MRP
Cyclophosphamide hydrate is a DNA alkylating agent, an inhibitor of DNA synthesis. Cyclophosphamide hydrate has antitumor and immunosuppressive activities.
T2863 P-Coumaric acid para-Coumaric Acid,4-Hydroxycinnamic acid,trans-4-Hydroxycinnamic acid,Trans-p-Coumaric acid,4-Coumaric acid,P-Hydroxycinnamic acid Endogenous Metabolite , Antibiotic
p-Coumaric acid (para-Coumaric Acid) is the abundant isomer of cinnamic acid, with antitumor and anti-mutagenic activities.
T2997 Rhein Rheinic Acid,Monorhein,NSC 38629,Rheic Acid,Rhubarb yellow Reactive Oxygen Species , Antibacterial , Autophagy
Rhein (NSC 38629) is an anthraquinone compound extracted from Polygonaceae Rheum Officinale with anti-inflammation and antitumor activities.
TN1190 14,15 β-Dihydroxyklaineanone 14,15beta-Dihydroxyklaineanone Parasite
14,15 β-Dihydroxyklaineanone(14,15beta-Dihydroxyklaineanone) is a bittersweet compound isolated from Eurycoma longifolia with antitumor-promoting, antischistosomal and plasmodium-killing activities.
T2853 Curcumol (-)-Curcumol Apoptosis , JAK
Curcumol ((-)-Curcumol), a pure monomer isolated extracted from Rhizoma Curcumaeis, has antitumor activities.
T7470 6-Chloropurine 6-Chloro-9H-purine Others
6-Chloropurine (6-Chloro-9H-purine) is a building block in chemical synthesis,with Antitumor activities.
T0876 Clioquinol Chinoform,Iodochlorhydroxyquin Mitophagy , Antibiotic , Autophagy , Antifungal
Clioquinol (Iodochlorhydroxyquin) is an orally bioavailable, lipophilic, copper-binding, halogenated 8-hydroxyquinoline with antifungal, antiparasitic and potential antitumor activities.

Compounds

Ganoderic acid F
T11363
Synonym:
Target: Others
S-trityl-L-Cysteine
T36816
Synonym: STLC
Target: Kinesin
CCT 031374 hydrobromide
T21685
Synonym:
Target: Wnt/beta-catenin
Antitumor agent-21
T3389
Synonym: TRX818
Target: Others
WAY-620645
T9991
Synonym:
Target: cholecystokinin
Protein kinase G inhibitor-2
T9940
Synonym:
Target: Others
Tiomolibdate diammonium
T19668
Synonym: Ammonium molybdenum sulfide,Ammonium tetrathiomolybdate,NSC 286644,ATTM,Coprexa
Target: Others
Dioscin
T6473
Synonym: CCRIS 4123,Collettiside III,Saponin
Target: Apoptosis, Autophagy
CBS9106
T14885
Synonym: SL-801
Target: CRM1
RKI-1447
T1898
Synonym: RKI1447
Target: ROCK
Menin-MLL inhibitor 20
T9399
Synonym:
Target: Epigenetic Reader Domain, Histone Methyltransferase
Ursolic acid acetate
T3819
Synonym: Acetylursolic acid,3-Acetylursolic Acid
Target: AChE
Sirtuin modulator 2
T9999
Synonym: N-(3-(imidazo[2,1-b]thiazol-6-yl)phenyl)-2-methoxybenzamide
Target: Others, Sirtuin
Cyclophosphamide hydrate
T0707
Synonym: Cyclophosphamide monohydrate
Target: DNA Alkylator/Crosslinker, DNA, MRP
p-Coumaric acid
T2863
Synonym: para-Coumaric Acid,4-Hydroxycinnamic acid,trans-4-Hydroxycinnamic acid,Trans-p-Coumaric acid,4-Coumaric acid,P-Hydroxycinnamic acid
Target: Endogenous Metabolite, Antibiotic
Rhein
T2997
Synonym: Rheinic Acid,Monorhein,NSC 38629,Rheic Acid,Rhubarb yellow
Target: Reactive Oxygen Species, Antibacterial, Autophagy
14,15 β-Dihydroxyklaineanone
TN1190
Synonym: 14,15beta-Dihydroxyklaineanone
Target: Parasite
Curcumol
T2853
Synonym: (-)-Curcumol
Target: Apoptosis, JAK
6-Chloropurine
T7470
Synonym: 6-Chloro-9H-purine
Target: Others
Clioquinol
T0876
Synonym: Chinoform,Iodochlorhydroxyquin
Target: Mitophagy, Antibiotic, Autophagy, Antifungal
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TargetMol